The authors reviewed current literature and curriculum resources on psychopharmacology and social work. They argue that baccalaureate and master of social work courses need to routinely include more in-depth knowledge on psychopharmacology and provide a more critical social work-focused approach to this content due to the increasing complexity of social work practice, including a knowledge explosion in the neurosciences. Toward this end, 7 curriculum modules are proposed, including suggestions for class activities and assignments and application of module content to field courses.